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Tagrisso

N-[2-[2-(dimethylamino)ethyl-methylamino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]prop-2-enamide · also: osimertinib, Mereletinib, osimertinibum, Osimertinib mesylate, osimertinib mesilate, Tyrosine Kinase Inhibitor - Ns

FormulaC28H33N7O2
Mol. weight499.619
PubChem CID71496458
InChIKeyDUYJMQONPNNFPI-UHFFFAOYSA-N
SMILESCN1C=C(C2=CC=CC=C21)C3=NC(=NC=C3)NC4=C(C=C(C(=C4)NC(=O)C=C)N(C)CCN(C)C)OC
10,065Patents
1,794Research papers
4,882Patents - last 3 years
558Papers - last 3 years

Who owns the IP

The organizations most actively patenting around this compound, ranked by referenced patent volume.

#AssigneePatents
1Gilead Sciences Inc204
2Bayer AG174
3Dana Farber Cancer Institute Inc129
4Bayer Pharma AG118
5AstraZeneca AB114
6Foundation Medicine Inc102
7Boehringer Ingelheim International GmbH101
8Kymera Therapeutics Inc94
9Institut National de la Santé et de la Recherche Médicale91
10F Hoffmann La Roche AG87

Explore the full landscape

This preview shows the leading assignees. Cypris reveals the full ownership landscape - every filing entity, filing trends, and portfolio momentum.

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Where innovation is concentrated

Patent classifications ranked by volume reveal the technical domains with the most active filing.

#CodeAreaPatents
1A61PTherapeutic activity (drug indications)8,379
2A61KMedicinal preparations8,050
3C07DHeterocyclic compounds4,482
4C07KPeptides2,449
5C12NMicroorganisms, enzymes971
6C12QMeasuring/testing involving enzymes872
7G01NInvestigating / analysing materials796
8C07BGeneral methods of organic chemistry618
9C07FOrganometallic compounds518
10Y02AClimate change adaptation390

AI mapped opportunity space

This preview shows where patent activity concentrates. Cypris maps the full classification landscape to surface technical whitespace and IP headroom.

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Most-cited patents

Patents ranked by forward citations reveal the foundational inventions the field continues to build on.

TitleYearAssigneeCited by
IMPROVED PROCESS FOR THE PREPARATION OF OSIMERTINIB (AZD9291) OR A SALT THEREOF, AND "AZD9291 ANILINE" OR A SALT THEREOF2017AstraZeneca AB11
A kind of Osimertinib preparation method2017JIANGSU SIMCERE PHARMACEUTICAL CO., LTD.7
OSIMERTINIB FOR USE IN THE TREATMENT OF NON-SMALL CELL LUNG CANCER2019AstraZeneca AB4
AN IMPROVED PROCESS FOR THE PREPARATION OF OSIMERTINIB MESYLATE2021Natco Pharma Ltd3
Anticancer compound osimertinib and synthesis method thereof2016HUANG YANGE2

Where research is gaining momentum

Research themes ranked by publication activity show where scientific interest is accelerating around this compound.

#Research topicPapers
1Lung Cancer Treatments and Mutations6
2Cancer Genomics and Diagnostics1
3Epigenetics and DNA Methylation1
4Extracellular vesicles in disease1
5Quinazolinone synthesis and applications1

Who's driving the science

The most-published authors working with this compound, alongside their primary affiliations.

#AuthorAffiliationPapers
1Suresh S. RamalingamEmory University27
2Myung‐Ju AhnSamsung Medical Center24
3James Chih‐Hsin YangNational Taiwan University Hospital21
4Yi‐Long WuGuangdong Academy of Medical Sciences21
5Byoung Chul ChoYonsei University19
6Helena A. YuMemorial Sloan Kettering Cancer Center15
7Pasi A. JänneDana-Farber Cancer Institute15
8Terufumi KatoKanagawa Prefectural Hospital Organization13
9Jia WangShanghai Innovative Research Center of Traditional Chinese Medicine6
10Yong HeDaping Hospital12

Research leaders

This preview lists the top authors. Cypris surfaces the full researcher landscape, their affiliations, and how scientific influence is shifting.

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The literature that defines it

The most-cited papers anchoring the scientific record for this compound.

Frequently asked questions

Common questions about this compound's patent and research landscape, answered from the underlying data.

What is the molecular formula and weight of Tagrisso?

Tagrisso has the molecular formula C28H33N7O2 and a molecular weight of 499.619 g/mol.

Which organizations hold the most patents related to Tagrisso?

Gilead Sciences Inc leads with 205 patents, followed by Bayer AG with 174 patents, and Dana Farber Cancer Institute Inc with 129 patents. Other significant patent holders include Bayer Pharma AG, AstraZeneca AB, and Foundation Medicine Inc.

What are the main research topics associated with Tagrisso in the literature?

The primary research focus is Lung Cancer Treatments and Mutations, with additional work in Cancer Genomics and Diagnostics, and Quinazolinone synthesis and applications.

Which researchers have published the most papers on Tagrisso?

Suresh S. Ramalingam from Emory University has published 27 papers, followed by Myung‐Ju Ahn from Samsung Medical Center with 24 papers, and James Chih‐Hsin Yang from National Taiwan University Hospital with 21 papers.

What does the patent trend show for Tagrisso-related inventions in recent years?

Patent filings show significant growth, with 712 patents in 2021 rising to 2,145 in 2023 and 2,253 in 2024. The last three years (2022–2024) account for 6,320 patents out of the total 10,065 patents in the database.

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