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miransertib

3-[3-[4-(1-aminocyclobutyl)phenyl]-5-phenylimidazo[4,5-b]pyridin-2-yl]pyridin-2-amine · also: miransertibum, Miransertib hydrochloride

FormulaC27H24N6
Mol. weight432.531
PubChem CID53262401
InChIKeyHNFMVVHMKGFCMB-UHFFFAOYSA-N
SMILESC1CC(C1)(C2=CC=C(C=C2)N3C4=C(C=CC(=N4)C5=CC=CC=C5)N=C3C6=C(N=CC=C6)N)N
2,818Patents
28Research papers
571Patents - last 3 years
2Papers - last 3 years

Who owns the IP

The organizations most actively patenting around this compound, ranked by referenced patent volume.

#AssigneePatents
1Janssen Pharmaceutica NV127
2Gilead Sciences Inc105
3Amgen Inc52
4Arcus Biosciences Inc47
5Merck Sharp & Dohme LLC47
6C4 Therapeutics Inc43
7Shanghai Hengrui Pharmaceutical Co Ltd35
8Scorpion Therapeutics Inc32
9Jiangsu Hengrui Medicine Co Ltd31
10Arqule Inc30

Explore the full landscape

This preview shows the leading assignees. Cypris reveals the full ownership landscape - every filing entity, filing trends, and portfolio momentum.

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Where innovation is concentrated

Patent classifications ranked by volume reveal the technical domains with the most active filing.

#CodeAreaPatents
1A61PTherapeutic activity (drug indications)2,203
2C07DHeterocyclic compounds2,036
3A61KMedicinal preparations1,768
4C07CAcyclic and carbocyclic compounds360
5C07KPeptides280
6C07HSugars and derivatives199
7C07FOrganometallic compounds198
8C07BGeneral methods of organic chemistry160
9Y02PClimate change mitigation: production145
10C12NMicroorganisms, enzymes134

AI mapped opportunity space

This preview shows where patent activity concentrates. Cypris maps the full classification landscape to surface technical whitespace and IP headroom.

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Where research is gaining momentum

Research themes ranked by publication activity show where scientific interest is accelerating around this compound.

#Research topicPapers
1PI3K/AKT/mTOR signaling in cancer1

Who's driving the science

The most-published authors working with this compound, alongside their primary affiliations.

#AuthorAffiliationPapers
1Brian SchwartzArqule (United States)10
2Giovanni AbbadessaArqule (United States)7
3Yi YuArqule (United States)7
4Leslie G. BieseckerNational Human Genome Research Institute4
5Carlotta RanieriUniversity of Bari Aldo Moro3
6Kimloan NguyenNational Center for Advancing Translational Sciences3
7Kyeong Ri YuNational Center for Advancing Translational Sciences3
8Pranav ShahNational Center for Advancing Translational Sciences3
9Ronald E. SavageArqule (United States)3
10Xin XuNational Center for Advancing Translational Sciences3

Research leaders

This preview lists the top authors. Cypris surfaces the full researcher landscape, their affiliations, and how scientific influence is shifting.

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The literature that defines it

The most-cited papers anchoring the scientific record for this compound.

Frequently asked questions

Common questions about this compound's patent and research landscape, answered from the underlying data.

What is the molecular formula and weight of miransertib?

Miransertib has the molecular formula C27H24N6 and a molecular weight of 432.531 g/mol. Its IUPAC name is 3-[3-[4-(1-aminocyclobutyl)phenyl]-5-phenylimidazo[4,5-b]pyridin-2-yl]pyridin-2-amine.

Which companies hold the most patents related to miransertib?

Janssen Pharmaceutica NV leads with 127 patents, followed by Gilead Sciences Inc with 105 patents, and Amgen Inc with 52 patents. Other significant patent holders include Arcus Biosciences Inc and Merck Sharp and Dohme LLC, each with 47 patents.

What are the primary research areas associated with miransertib publications?

Published research on miransertib focuses on several key areas: targeting the PI3K/AKT pathway as an allosteric AKT inhibitor, treatment of Proteus Syndrome, efficacy in PIK3CA-related overgrowth spectrum disorders, and clinical applications in PIK3CA-related overgrowth syndrome in pediatric patients.

Who are the leading researchers publishing on miransertib and their affiliations?

Brian Schwartz from Arqule (United States) is the most prolific author with 10 papers on miransertib. Other significant contributors include Giovanni Abbadessa and Yi Yu from Arqule (7 papers each), and Leslie G. Biesecker from the National Human Genome Research Institute (4 papers).

What is the recent patent filing trend for miransertib-related technology?

Patent filing activity shows strong growth, with 287 patents filed in 2024 and 235 in 2023, representing the highest annual filing rates in the tracked period. In the last three years, 578 patents have been filed related to miransertib technology.

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